Synthesis and biological activities of novel quinazolinone derivatives containing a 1,2,4-triazolylthioether moiety

References

Asker, F.W., Abbas, S. A. R., Al-Bayati, R. I., & Al-Tamemi, H.A. (2014). Synthesis and biological evaluation of new quinazolinone derivatives. European Journal of Chemistry, 5, 628–634. DOI: 10.5155/eurjchem.5.4.628-634.112010.5155/eurjchem.5.4.628-634.1120Search in Google Scholar

Bartroli, J., Tumo, E., Algueró, M., Boncompte, E., Vericat, M. L., Conte, L., Ramis, J., Merlos, M., Garcia-Rafanell, J., & Forn, J. (1998). New azole antifungals. 3. Synthesis and antifungal activity of 3-substituted-4(3H)-quinazolinones. Journal of Medicinal Chemistry, 41, 1869–1882. DOI: 10.1021/jm9707277.10.1021/jm9707277Search in Google Scholar PubMed

Cao, S. L., Feng, Y. P., Jiang, Y. Y., Liu, S. Y., Ding, G. Y., & Li, R. T. (2005). Synthesis and in vitro antitumor activity of4(3H)-quinazolinone derivatives with dithiocarbamate sidechains. Bioorganic & Medicinal Chemistry Letters, 15, 1915–1917. DOI: 10.1016/j.bmcl.2005.01.083.10.1016/j.bmcl.2005.01.083Search in Google Scholar PubMed

Cao, X. F., Li, F., Hu, M., Lu, W. C., Yu, G. A., & Liu, S. H.(2008). Chiral γ-Aryl-1H-1,2,4-triazole derivatives as highlypotential antifungal agents: Design, synthesis, structure andin vitro fungicidal activities. Journal of Agricultural andFood Chemistry, 56, 11367–11375. DOI: 10.1021/jf8026843.10.1021/jf8026843Search in Google Scholar PubMed

Dixit, R., Mehta, H., & Dixit, B. (2015). Synthesis, characterization and antimicrobial studies of new 2-(2-chloroquinolin-3-yl)-3-(substituted phenyl/pyridinyl) quinazolin-4(3H)-onederivatives using L-proline as a catalyst. Medicinal Chemistry Research, 24, 773–786. DOI: 10.1007/s00044-014-1116-810.1007/s00044-014-1116-8Search in Google Scholar

El-Hashash, M. A., Elshahawi, M. M., Ragab, E. A., & Nagdy, S. (2015). Synthesis and antifungal activity of novelquinazolin-4(3H)-one derivatives. Synthetic Communications,45, 2240–2250. DOI: 10.1080/00397911.2015.1074697.10.1080/00397911.2015.1074697Search in Google Scholar

Gülerman, N. N., Doğan, H. N., Rollas, S., Johansson, C.,& Çelik, C. (2001). Synthesis and structure elucidation of some new thioether derivatives of 1,2,4-triazoline-3-thiones and their antimicrobial activities. II Farmaco, 56, 953–958.DOI: 10.1016/s0014-827x(01)01167-3.10.1016/s0014-827x(01)01167-3Search in Google Scholar PubMed

Hasan, A., Francis, N., Thomas, N. F., & Gapil, S. (2011).Synthesis, characterization and antifungal evaluation of 5-substituted-4-amino-1,2,4-triazole-3-thioesters. Molecules,16, 1297–1309. DOI: 10.3390/molecules16021297.10.3390/molecules16021297Search in Google Scholar PubMed PubMed Central

Holla, B. S., Gonsalves, R., & Shenoy, S. (2000). Synthesis and antibacterial studies of a new series of 1,2-bis(1,3,4-oxadiazol-2-yl)ethanes and 1,2-bis(4-amino-1,2,4-triazol-3-yl)ethanes.European Journal of Medicinal Chemistry, 35, 267–271.DOI: 10.1016/s0223-5234(00)00154-9.10.1016/s0223-5234(00)00154-9Search in Google Scholar PubMed

Jatav, V., Mishra, P., Kashaw, S., & Stables, J. P. (2008). CNS depressant and anticonvulsant activities of some novel 3-[5-substituted-1,3,4-thiadiazole-2-yl]-2-styryl-quinazoline-4(3H)-ones. European Journal of Medicinal Chemistry, 43,1945–1954. DOI: 10.1016/j.ejmech.2007.12.003.10.1016/j.ejmech.2007.12.003Search in Google Scholar PubMed

Liu, F., Luo, X. Q., Song, B. A., Bhadury, P. S., Yang, S., Jin, L. H., Xue, W., & Hu, D. Y. (2008). Synthesis and antifungal activity of novel sulfoxide derivatives containing trimethoxyphenyl substituted 1,3,4-thiadiazole and 1,3,4-oxadiazole moiety. Bioorganic & Medicinal Chemistry, 16, 3632–3640. DOI: 10.1016/j.bmc.2008.02.006.10.1016/j.bmc.2008.02.006Search in Google Scholar PubMed

Liu, J. H., Liu, Y., Jian, J. Y., & Bao, X. P. (2013). Synthesis and fungicidal activities of novel quinazoline derivatives containing 1,2,4-triazole Schiff-base unit. Chinese Journal of Organic Chemistry, 33, 370–374. DOI: 10.6023/cjoc201209023.10.6023/cjoc201209023Search in Google Scholar

Ma, J., Li, P., Li, X. Y., Shi, Q. C., Wan, Z. H., Hu, D. Y., Jin, L. H., & Song, B. A. (2014). Synthesis and antiviral bioactivity of novel 3-((2-((1E,4E)-3-oxo-5-arylpenta-1,4-dien-1-yl)phenoxy)methyl)-4(3H)-quinazolinone derivatives. Journal of Agricultural and Food Chemistry, 62, 8928–8934. DOI: 10.1021/jf502162y.10.1021/jf502162ySearch in Google Scholar PubMed

Mali, J. R., Pratap, U. R., Netankar, P. D., & Mane, R. A. (2009). An efficient synthetic route for quinazolinyl 4-thiazolidinones. Tetrahedron Letters, 50, 5025–5027. DOI: 10.1016/j.tetlet.2009.06.086.10.1016/j.tetlet.2009.06.086Search in Google Scholar

Panneerselvam, P., Rather, B. A., Reddy, D. R. S., & Kumar, N. R. (2009). Synthesis and anti-microbial screening of some Schiff bases of 3-amino-6,8-dibromo-2-phenylquinazolin-4 (3H)-ones. European Journal of Medicinal Chemistry, 44, 2328–2333. DOI: 10.1016/j.ejmech.2008.04.010.10.1016/j.ejmech.2008.04.010Search in Google Scholar PubMed

Patil, B. S., Krishnamurthy, G., Naik, H. S. B., Latthe, P. R., & Ghate, M. (2010). Synthesis, characterization and antimicrobial studies of 2-(4-methoxy-phenyl)-5-methyl-4-(2-arylsulfanyl-ethyl)-2,4-dihydro-[1,2,4]triazolo-3-ones and their corresponding sulfones. European Journal of Medicinal Chemistry, 45, 3329–3334. DOI: 10.1016/j.ejmech.2010.04. 016.10.1016/j.ejmech.2010.04.016Search in Google Scholar PubMed

Plech, T., Wujec, M., Kosikowska, U., & Malm, A. (2013). Synthesis and antibacterial activity of 4,5-disubstituted-1,2,4-triazole-3-thiones. Letters in Drug Design & Discovery, 10, 917–922. DOI: 10.2174/15701808113109990082.10.2174/15701808113109990082Search in Google Scholar

Shi, L. P., Jiang, K. M., Jiang, J. J., Jin, Y., Tao, Y. H., Li, K., Wang, X. H., & Lin, J. (2013). Synthesis and antimicrobial activity of polyhalobenzonitrile quinazolin-4(3H)-one derivatives. Bioorganic & Medicinal Chemistry Letters, 23, 5958–5963. DOI: 10.1016/j.bmcl.2013.08.068.10.1016/j.bmcl.2013.08.068Search in Google Scholar PubMed

Shin, K. J., Koo, K. D., Yoo, K. H., Kang, Y. K., Park, S.W., & Kim, D. J. (2001). Synthesis and biological properties of new 1-β-methylcarbapenems containing heteroaromatic thioether moiety. Bioorganic & Medicinal Chemistry Letters, 11, 2397– 2399. DOI: 10.1016/s0960-894x(01)00451-6.10.1016/s0960-894x(01)00451-6Search in Google Scholar PubMed

Sun, J., Li, D. D., Li, J. R., Fang, F., Du, Q. R., Qian, Y., & Zhu, H. L. (2013). Design, synthesis, biological evaluation and molecular modeling study of 4-alkoxyquinazoline derivatives as potential VEGFR2 kinase inhibitors. Organic & Biomolecular Chemistry, 11, 7676–7686. DOI: 10.1039/c3ob41136b.10.1039/c3ob41136bSearch in Google Scholar PubMed

Turan-Zitouni, G., Kaplancikli, Z. A., Yildiz, M. T., Chevallet, P., & Kaya, D. (2005). Synthesis and antimicrobial activity of 4-phenyl/cyclohexyl-5-(1-phenoxyethyl)-3-[N-(2-thiazolyl)acetamido]thio-4H-1,2,4-triazole derivatives. European Journal of Medicinal Chemistry, 40, 607–613. DOI: 10.1016/j.ejmech.2005.01.007.10.1016/j.ejmech.2005.01.007Search in Google Scholar PubMed

Wang, X., Li, P., Li, Z. N., Yin, J. A., He, M., Xue, W., Chen, Z. W., & Song, B. A. (2013). Synthesis and bioactivity evaluation of novel arylimines containing a 3-aminoethyl-2-[(ptrifluoromethoxy) anilino]-4(3H)-quinazolinone moiety. Journal of Agricultural and Food Chemistry, 61, 9575–9582. DOI: 10.1021/jf403193q.10.1021/jf403193qSearch in Google Scholar PubMed

Xu, W. M., Han, F. F., He, M., Hu, D. Y., He, J., Yang, S., & Song, B. A. (2012). Inhibition of tobacco bacterial wilt with sulfone derivatives containing an 1,3,4-oxadiazole moiety. Journal of Agricultural and Food Chemistry, 60, 1036– 1041. DOI: 10.1021/jf203772d10.1021/jf203772dSearch in Google Scholar PubMed

Zhang, F., Wen, Q., Wang, S. F., Karim, B. S., Yang, Y. S., Liu, J. J., Zhang, W. M., & Zhu, H. L. (2014). Design, synthesis and antibacterial activities of 5-(pyrazin-2-yl)-4H-1,2,4-triazole-3-thiol derivatives containing Schiff base formation as FabH inhibitory. Bioorganic & Medicinal Chemistry Letters, 24, 90–95. DOI: 10.1016/j.bmcl.2013.11.079.10.1016/j.bmcl.2013.11.079Search in Google Scholar PubMed

Zhu, S. R., Wang, J., Chandrashekar, G., Smith, E., Liu, X. J., & Zhang, Y. S. (2010). Synthesis and evaluation of 4-quinazolinone compounds as potential antimalarial agents. European Journal of Medicinal Chemistry, 45, 3864–3869. DOI: 10.1016/j.ejmech.2010.05.040.10.1016/j.ejmech.2010.05.040Search in Google Scholar PubMed PubMed Central