Skip to main content
Article Publicly Available

Medicinal Chemistry in Drug Discovery, India

Published/Copyright: November 18, 2014
Become an author with De Gruyter Brill

The increase in Medicinal Chemistry and Drug Discovery employment in Indian and Southeast Asian pharmaceutical companies and in the Contract Research Organizations collaborating with US and European companies has created a need for chemists and drug discovery scientists to acquire state-of-the-art knowledge of medicinal chemistry and other drug discovery areas. This course will emphasize the design strategy that takes into account drug metabolism and pharmacokinetics (DMPK), and toxicophore. The course will be based on the successful first year program in 2013 and the Drew University Residential School on Medicinal Chemistry, taught annually since 1986 on the Drew University campus in Madison, New Jersey. MCI 2015 will comprise 4.5 days of content, including 18-20 1-hour lectures on topics covering all aspects of medicinal chemistry from target selection and validatation, to hit identification, hit-to-lead chemistry, and lead optimization. New lectures on preclinical toxicity and clinical development will be added for the 2015 program. Four case history presentations of successful drug discovery programs will also be included. The course will be taught mainly by faculty from the US, with some local Indian faculty members also participating. The plan is to increase the number of Indian faculty members in subsequent years. The performance and value of the course will be assessed after the end of the three-year period, and a decision whether to continue in the same format made at that time. The desired outcome will be to enroll 80-100 attendees each year, and provide them with a strong introduction to the practice of medicinal chemistry in drug discovery. We are actively seeking the participation of other emerging or developing countries such as Singapore, Malaysia, South Africa, etc.

Following the success of the four-day Residential Course in Medicinal Chemistry (see Chem Int, March 2014, p.20), the current program is designed to educate drug discovery and early clinical development scientists from industry and academia, including the areas of medicinal chemistry, formulation chemistry, metabolism, and toxicology, on the importance of interplay among the different areas and their team efforts to execute a successful drug discovery and development process. The next Course is planned for February 2015.

For more information, contact the Task Group Chair Balu Balasubramanian <>

www.iupac.org/project/2014-011-2-700

Online erschienen: 2014-11-18
Erschienen im Druck: 2014-11-1

©2014 by Walter de Gruyter Berlin/Boston

Articles in the same Issue

  1. Masthead - Full issue pdf
  2. From the Editor
  3. Contents
  4. Features
  5. Planetary Boundaries and Chemical Pollution: A Grail Quest?
  6. Research Integrity: Science Community Needs to Address Threats by Research Assessments
  7. IUPAC and ICSU—A Comment
  8. Invitation to host the ICSU Secretariat for the Committee on Freedom and Responsibility in the conduct of Science (CFRS)
  9. Drug Design and Development: A Research Center More Than Twenty Years in the Making
  10. Youth Views on Sustainability: Size Matters, But So Does Speed
  11. IUPAC Wire
  12. Mort Hoffman Receives Chemistry Education Award
  13. Vânia G. Zuin is awarded the CHEMRAWN VII Prize for Atmospheric and Green Chemistry
  14. Sébastien Perrier received the 2014 IUPAC- Samsung Young Polymer Scientist Award
  15. DSM Materials Sciences Award 2014 goes to Prof. Jian Ping Gong
  16. 2015 IUPAC-SOLVAY International Award for Young Chemists announced
  17. In Memoriam: Gerrit den Boef
  18. The Project Place
  19. Critically evaluated rate parameters for chain-length-dependent termination in radical polymerization of styrene and n-alkyl methacrylates
  20. Guidelines for assigning values and calculating uncertainties to the standard atomic weights
  21. Nano-pesticides in the Environment
  22. Medicinal Chemistry in Drug Discovery, India
  23. Biological Context by TextData-mining
  24. IUPAC Recommendations for the definition, preferred symbol for all transport properties
  25. End-of-line hyphenation of systematic chemical names
  26. Making an imPACt
  27. Single-molecule fluorescence imaging by total internal reflection fluorescence microscopy (IUPAC Technical Report)
  28. Updates to the International System of Units (SI) brochure (8th edition)
  29. Variation in the terrestrial isotopic composition and atomic weight of argon (IUPAC Technical Report)
  30. Provisional Recommendations
  31. Nomenclature and Graphic Representations for Chemically Modified Polymers
  32. Conference Call
  33. Big Data for International Scientific Programmes
  34. CD3—A Celebration More Than 20 Years in the Making
  35. Solid State Chemistry
  36. Where 2B & Y
  37. Highlights in Medicinal Chemistry
  38. European Polymer Congress
  39. Point of Care Testing
  40. Research Integrity
  41. Mark Your Calendar
  42. Index 2014
  43. Stamps International
  44. The International Year of Crystallography (2014): A Philatelic Celebration
Downloaded on 16.4.2026 from https://www.degruyterbrill.com/document/doi/10.1515/ci-2014-0618/html
Scroll to top button